SCHEMBL6971189

SCHEMBL6971189

COc1ccc(NC(=O)c2c[c]ccc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 11/20 0.68
RAB9A P51151 11/20 0.68
SMN1; SMN2 Q16637 4/20 0.64
TP53 P04637 3/20 0.64
ALOX15 P16050 1/20 0.64
CASP3 P42574 1/20 0.56
SENP7 Q9BQF6 1/20 0.56
KDM4E B2RXH2 3/20 0.54
ALDH1A1 P00352 3/20 0.54
CYP1A2 P05177 2/20 0.54
KCNK9 Q9NPC2 1/20 0.54
MAPT P10636 1/20 0.53
KMT2A Q03164 4/20 0.52
MEN1 O00255 3/20 0.52
GAA P10253 2/20 0.52
TSHR P16473 1/20 0.52
NFKB1 P19838 1/20 0.52
NFKB2 Q00653 1/20 0.52
RELA Q04206 1/20 0.52
TAS1R3 Q7RTX0 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5465598 0.85 RAB9A (0.64) NPC1RAB9ASMN1; SMN2TP53ALOX15
SCHEMBL5461596 0.82 NPC1 (0.60) NPC1RAB9ASMN1; SMN2TP53CASP3
SCHEMBL483328 0.81 RAB9A (0.77) NPC1RAB9ASMN1; SMN2TP53ALOX15
SCHEMBL4963650 0.81 RAB9A (1.00) NPC1RAB9ASMN1; SMN2TP53ALOX15
SCHEMBL750970 0.81 SIRT1 (0.58) NPC1RAB9ASMN1; SMN2KDM4EKCNK9
SCHEMBL7573916 0.80 MAPK1 (0.53) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL5474341 0.80 KMT2A (0.63) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL27931870 0.80 POLB (0.61) NPC1RAB9ASMN1; SMN2TP53KDM4E
Iodide SCHEMBL30758596 0.80 RAB9A (0.97) NPC1RAB9ASMN1; SMN2TP53ALOX15
Hydrochloric Acid SCHEMBL29693066 0.80 RAB9A (0.97) NPC1RAB9ASMN1; SMN2TP53ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed