Proxyfan

Proxyfan

SCHEMBL15929504

c1ccc(COCCCc2cnc[nH]2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 1.00
HRH4 Q9H3N8 5/20 1.00
TAAR1 Q96RJ0 1/20 0.61
KCNH2 Q12809 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Proxyfan SCHEMBL29462311 0.93 HRH3 (0.87) HRH3HRH4
SCHEMBL2536900 0.80 HRH3 (0.93) HRH3HRH4TAAR1
SCHEMBL224745 0.77 TAAR1 (1.00) HRH3HRH4TAAR1
SCHEMBL194703 0.75 HRH3 (0.71) HRH3HRH4
SCHEMBL4069939 0.74 TDP1 (0.64) HRH3HRH4
SCHEMBL4217229 0.73 HRH3 (0.58) HRH3HRH4
SCHEMBL4769249 0.73 HRH4 (0.57) HRH3HRH4
SCHEMBL18536735 0.72 HRH3 (0.57) HRH3HRH4TAAR1
SCHEMBL2741614 0.72 ADRA1A (0.68) HRH3HRH4TAAR1
SCHEMBL8964986 0.72 HRH3 (0.79) HRH3HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10449144-B2 WT1 peptide cancer vaccine composition for transdermal administration NITTO DENKO CORPORATION (JP) 2019-10-22 US disclosed
US-10206985-B2 WT1 peptide cancer vaccine composition for mucosal administration NITTO DENKO CORPORATION (JP) 2019-02-19 US disclosed
US-10195258-B2 Tape preparation of WT1 peptide cancer vaccine for transdermal administration NITTO DENKO CORPORATION (JP) 2019-02-05 US disclosed
US-20170224813-A1 VACCINE PHARMACEUTICAL COMPOSITION FOR SUPPRESSING APOPTOSIS OF CTL OR INHIBITING SUPPRESSION OF INDUCTION OF CTL NITTO DENKO CORPORATION (JP) 2017-08-10 US disclosed
US-20150080380-A1 Therapeutic Uses GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2015-03-19 US disclosed
US-20150080380-A1 Therapeutic Uses GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2015-03-19 US disclosed
US-20140220079-A1 VACCINE COMPOSITION FOR MUCOSAL ADMINISTRATION NITTO DENKO CORPORATION (JP) 2014-08-07 US disclosed
US-20140220058-A1 VACCINE COMPOSITION FOR TRANSDERMAL OR MUCOSAL ADMINISTRATION NITTO DENKO CORPORATION (JP) 2014-08-07 US disclosed
US-20140220063-A1 VACCINE COMPOSITION NITTO DENKO CORPORATION (JP) 2014-08-07 US disclosed
US-20140220100-A1 VACCINE COMPOSITION FOR TRANSDERMAL ADMINISTRATION NITTO DENKO CORPORATION (JP) 2014-08-07 US disclosed
US-20140220059-A1 WT1 PEPTIDE CANCER VACCINE COMPOSITION FOR MUCOSAL ADMINISTRATION INTERNATIONAL INSTITUTE OF CANCER IMMUNOLOGY, INC. (JP) 2014-08-07 US disclosed
US-20140220105-A1 TAPE PREPARATION OF WT1 PEPTIDE CANCER VACCINE FOR TRANSDERMAL ADMINISTRATION INTERNATIONAL INSTITUTE OF CANCER IMMUNOLOGY, INC. (JP) 2014-08-07 US disclosed
US-20140220055-A1 WT1 PEPTIDE CANCER VACCINE COMPOSITION FOR TRANSDERMAL ADMINISTRATION INTERNATIONAL INSTITUTE OF CANCER IMMUNOLOGY, INC. (JP) 2014-08-07 US disclosed
US-20140220057-A1 WT1 PEPTIDE CANCER VACCINE COMPOSITION FOR TRANSDERMAL ADMINISTRATION INTERNATIONAL INSTITUTE OF CANCER IMMUNOLOGY, INC. (JP) 2014-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (13 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140220105-A1 TAPE PREPARATION OF WT1 PEPTIDE CANCER VACCINE FOR TRANSDERMAL ADMINISTRATION TAP1, TAP2, MICA HRH3 4254/4885HRH4 4547/4885TAAR1 2767/4885
US-10206985-B2 WT1 peptide cancer vaccine composition for mucosal administration MUC1, TAP1, MICA HRH3 3667/4885HRH4 4151/4885TAAR1 3709/4885
US-10449144-B2 WT1 peptide cancer vaccine composition for transdermal administration TAP1, TAP2, MICA HRH3 3871/4885HRH4 4045/4885TAAR1 2639/4885
US-20140220057-A1 WT1 PEPTIDE CANCER VACCINE COMPOSITION FOR TRANSDERMAL ADMINISTRATION TAP1, TAP2, MUC1 HRH3 3261/4885HRH4 3271/4885TAAR1 2093/4885
US-20140220100-A1 VACCINE COMPOSITION FOR TRANSDERMAL ADMINISTRATION ERBB2, EGFR, ERBB3 HRH3 1087/4885HRH4 644/4885TAAR1 1901/4885
US-20140220058-A1 VACCINE COMPOSITION FOR TRANSDERMAL OR MUCOSAL ADMINISTRATION CD69, TSLP, MUC1 HRH3 369/4885HRH4 306/4885TAAR1 493/4885
US-10195258-B2 Tape preparation of WT1 peptide cancer vaccine for transdermal administration TAP1, TAP2, MICA HRH3 4254/4885HRH4 4547/4885TAAR1 2767/4885
US-20150080380-A1 Therapeutic Uses HRH3, HRH4, HRH2 HRH3 1/4885HRH4 2/4885TAAR1 190/4885
US-20140220055-A1 WT1 PEPTIDE CANCER VACCINE COMPOSITION FOR TRANSDERMAL ADMINISTRATION TAP1, TAP2, MICA HRH3 3871/4885HRH4 4045/4885TAAR1 2639/4885
US-20170224813-A1 VACCINE PHARMACEUTICAL COMPOSITION FOR SUPPRESSING APOPTOSIS OF CTL OR INHIBITING SUPPRESSION OF INDUCTION OF CTL BAX, GZMB, BCL2 HRH3 3284/4885HRH4 3713/4885TAAR1 4520/4885
US-20140220079-A1 VACCINE COMPOSITION FOR MUCOSAL ADMINISTRATION MUC1, ERBB2, TLR5 HRH3 486/4885HRH4 394/4885TAAR1 2673/4885
US-20140220059-A1 WT1 PEPTIDE CANCER VACCINE COMPOSITION FOR MUCOSAL ADMINISTRATION MUC1, TAP1, MICA HRH3 3667/4885HRH4 4151/4885TAAR1 3709/4885
US-20140220063-A1 VACCINE COMPOSITION MYD88, IRF3, CD14 HRH3 3420/4885HRH4 4295/4885TAAR1 4309/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.