SCHEMBL6972107

SCHEMBL6972107

CCOC(=O)CCN1C(=O)CCN(C(=O)c2ccc(N)cc2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.46
RAB9A P51151 3/20 0.45
NPC1 O15118 2/20 0.45
AVPR2 P30518 4/20 0.45
AVPR1A P37288 3/20 0.45
KMT2A Q03164 4/20 0.42
HPGD P15428 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MEN1 O00255 3/20 0.40
ALDH1A1 P00352 4/20 0.39
ALOX15 P16050 1/20 0.39
CNR2 P34972 2/20 0.39
POLB P06746 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAOA P21397 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6957126 0.94 NOTUM (0.44) NOTUMRAB9ANPC1AVPR2AVPR1A
SCHEMBL6960127 0.90 NPSR1 (0.49) NOTUMRAB9ANPC1AVPR2AVPR1A
SCHEMBL6969126 0.86 L3MBTL1 (0.45) NOTUMRAB9ANPC1KMT2AHPGD
SCHEMBL6967260 0.81 AVPR2 (0.48) NOTUMRAB9ANPC1AVPR2AVPR1A
SCHEMBL6970673 0.81 AVPR2 (0.48) RAB9ANPC1AVPR2AVPR1AKMT2A
SCHEMBL6969761 0.81 L3MBTL1 (0.43) NOTUMRAB9ANPC1KMT2ASMN1; SMN2
SCHEMBL6960448 0.80 AVPR2 (0.53) AVPR2AVPR1AOXTR
SCHEMBL6969600 0.79 AVPR2 (0.46) RAB9ANPC1AVPR2AVPR1AKMT2A
SCHEMBL6970661 0.79 ALDH1A1 (0.46) RAB9ANPC1AVPR2AVPR1AKMT2A
SCHEMBL6969459 0.79 ALDH1A1 (0.46) RAB9ANPC1AVPR2AVPR1AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed