SCHEMBL6969459

SCHEMBL6969459

CCOC(=O)CN1C(=O)CCN(C(=O)c2ccc(N)cc2)c2cc(C)ccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
KMT2A Q03164 3/20 0.43
RAB9A P51151 3/20 0.43
MEN1 O00255 2/20 0.43
LMNA P02545 5/20 0.42
NPSR1 Q6W5P4 2/20 0.40
USP2 O75604 1/20 0.39
HTT P42858 1/20 0.39
PPARG P37231 1/20 0.39
NPC1 O15118 2/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TP53 P04637 2/20 0.39
CYP1A2 P05177 2/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
AVPR2 P30518 1/20 0.37
AVPR1A P37288 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6970661 0.96 ALDH1A1 (0.46) ALDH1A1KMT2ARAB9AMEN1LMNA
SCHEMBL6969797 0.90 LMNA (0.44) ALDH1A1KMT2ARAB9AMEN1LMNA
SCHEMBL6960127 0.89 NPSR1 (0.49) ALDH1A1KMT2ARAB9AMEN1LMNA
SCHEMBL6966483 0.87 SMN1; SMN2 (0.44) ALDH1A1KMT2ARAB9AMEN1LMNA
SCHEMBL6969382 0.86 LMNA (0.55) ALDH1A1KMT2ARAB9AMEN1LMNA
SCHEMBL6962852 0.85 CA1 (0.43) ALDH1A1KMT2ARAB9AMEN1LMNA
SCHEMBL6968111 0.85 ALDH1A1 (0.43) ALDH1A1KMT2ARAB9AMEN1LMNA
SCHEMBL6967645 0.84 LOXL2 (0.40) ALDH1A1KMT2ARAB9AMEN1LMNA
SCHEMBL6972651 0.83 ALDH1A1 (0.41) ALDH1A1KMT2ARAB9AMEN1LMNA
SCHEMBL6971802 0.83 SMN1; SMN2 (0.44) ALDH1A1KMT2ARAB9AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed