SCHEMBL6972138

SCHEMBL6972138

Cc1n[nH]c(C)c1NC(c1ccccc1)c1cccc(C#N)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.39
PLK1 P53350 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
S1PR3 Q99500 2/20 0.35
HPGDS O60760 1/20 0.35
MAPK1 P28482 1/20 0.35
PIN1 Q13526 1/20 0.34
MAP4K4 O95819 1/20 0.34
GSK3A P49840 1/20 0.34
EP300 Q09472 2/20 0.34
SOS1 Q07889 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
GPR139 Q6DWJ6 1/20 0.33
CHEK1 O14757 1/20 0.33
AKT2 P31751 1/20 0.33
MGLL Q99685 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972370 0.71 S1PR1 (0.36) LRRK2PLK1SMN1; SMN2MAPK1PIN1
SCHEMBL22927647 0.66 HPGDS (0.42) SMN1; SMN2S1PR3HPGDSCNR1CNR2
SCHEMBL17069277 0.64 TSHR (0.48) CNR1CNR2GPR139SLC6A2SLC6A4
SCHEMBL17071849 0.64 TSHR (0.48) CNR1CNR2GPR139SLC6A2SLC6A4
SCHEMBL22927646 0.64 HPGDS (0.40) SMN1; SMN2S1PR3HPGDSCNR1CNR2
SCHEMBL28716544 0.64 HPGDS (0.40) SMN1; SMN2S1PR3HPGDSCNR1CNR2
SCHEMBL28716543 0.64 HPGDS (0.40) SMN1; SMN2S1PR3HPGDSCNR1CNR2
SCHEMBL24963400 0.63 CHEK1 (0.57) PIN1MAP4K4GSK3ACHEK1AKT2
SCHEMBL30239372 0.63 CHEK1 (0.57) PIN1MAP4K4GSK3ACHEK1AKT2
SCHEMBL17069276 0.62 TSHR (0.45) CNR1CNR2GPR139MGLLSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed