SCHEMBL30239372

SCHEMBL30239372

Cc1n[nH]c(C)c1-c1ccc(-c2cccc(C#N)c2)cc1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.57
AKT2 P31751 1/20 0.57
FASN P49327 1/20 0.47
PGR P06401 6/20 0.46
AR P10275 1/20 0.46
GSK3A P49840 2/20 0.45
MAP4K4 O95819 1/20 0.45
IDO1 P14902 2/20 0.44
MARK3 P27448 1/20 0.44
PIN1 Q13526 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
MKNK1 Q9BUB5 1/20 0.43
MAOB P27338 1/20 0.41
ACVR1 Q04771 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24963400 1.00 CHEK1 (0.57) CHEK1AKT2FASNPGRAR
SCHEMBL3074271 0.83 CHEK1 (0.59) CHEK1AKT2FASNMKNK1ACVR1
SCHEMBL7395177 0.78 IDO1 (0.46) FASNPGRARGSK3AMAP4K4
SCHEMBL16209719 0.76 AKT2 (0.79) CHEK1AKT2MKNK1ACVR1
SCHEMBL7430278 0.75 IDO1 (0.43) FASNPGRARGSK3AMAP4K4
SCHEMBL4443914 0.74 ALDH1A1 (0.52) PGRARMAP4K4CLK4
SCHEMBL7404293 0.74 F11 (0.52) FASNPGRGSK3AMAP4K4IDO1
SCHEMBL873114 0.74 AKT2 (1.00) CHEK1AKT2GSK3AMARK3MKNK1
SCHEMBL27787243 0.74 CLK4 (0.63) PGRMAP4K4IDO1CLK4MAOB
SCHEMBL5269506 0.73 L3MBTL1 (0.59) PGRGSK3AMAP4K4IDO1PIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023004280-A1 SELECTIVE PYRAZOLE LRRK2 INHIBITORS AND METHODS FOR USE THEREOF THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2023-01-26 WO claimed