SCHEMBL6972267

SCHEMBL6972267

CC(=O)c1c(-c2ncccn2)n[nH]c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
ALDH1A1 P00352 2/20 0.35
PDE4D Q08499 1/20 0.35
CSNK2A2 P19784 2/20 0.34
KDR P35968 2/20 0.34
CSNK2B P67870 2/20 0.34
CSNK2A1 P68400 2/20 0.34
TDP2 O95551 1/20 0.34
CCNE2 O96020 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
CSNK1A1 P48729 1/20 0.33
CSNK1D P48730 1/20 0.33
CLK2 P49760 1/20 0.33
CSNK1G1 Q9HCP0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13184233 0.74 DYRK1A (0.41) HSP90AA1NPC1GAAMAPTCYP3A4
SCHEMBL3229317 0.71 HCAR2 (0.37) CYP3A4MAPK1P2RX7KMT2A
SCHEMBL1640767 0.69 PDE4D (0.59) HSP90AA1HSP90AB1PDE4DCSNK2A2KDR
SCHEMBL10919855 0.68 PDE4D (0.45) ALDH1A1PDE4DTDP2SMN1; SMN2MAPT
SCHEMBL10923051 0.68 HSP90AA1 (0.41) HSP90AA1HSP90AB1ALDH1A1GAAMAPT
SCHEMBL29656885 0.64 ALDH1A1 (0.41) NPC1RAB9AALDH1A1TDP2SMN1; SMN2
SCHEMBL22498528 0.64 ALDH1A1 (0.41) NPC1RAB9AALDH1A1TDP2SMN1; SMN2
SCHEMBL4382163 0.63 RAB9A (0.49) HSP90AA1HSP90AB1RAB9AALDH1A1GAA
SCHEMBL12106580 0.63 CYP1A2 (0.39) ALDH1A1PDE4DCSNK2A2KDRCSNK2B
SCHEMBL12106575 0.63 PDE4D (0.43) HSP90AA1HSP90AB1ALDH1A1PDE4DCSNK2A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0784055-B1 PYRIMIDINYLPYRAZOLE DERIVATIVE DAIICHI SEIYAKU CO (JP) 2003-02-12 EP disclosed