SCHEMBL6972720

SCHEMBL6972720

Brc1[c]cccc1Cc1ccncc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 9/20 0.36
CYP11B2 P19099 9/20 0.36
CYP17A1 P05093 8/20 0.36
CYP19A1 P11511 5/20 0.36
CYP3A4 P08684 6/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HRH4 Q9H3N8 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLB P06746 1/20 0.33
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6978264 0.83 HTR2A (0.42) CYP3A4SMN1; SMN2ALDH1A1HSD17B10
SCHEMBL6982912 0.81 HRH4 (0.41) CYP11B1CYP11B2HRH4HRH3CYP1A2
SCHEMBL28550049 0.73 KMT2A (0.47) CYP11B1CYP11B2CYP17A1CYP19A1CYP3A4
SCHEMBL27306793 0.69
SCHEMBL455177 0.69
SCHEMBL16952915 0.69
SCHEMBL6978761 0.68 GPR55 (0.46)
SCHEMBL8182895 0.68 CYP11B1 (0.39) CYP11B1CYP11B2CYP17A1CYP19A1CYP3A4
SCHEMBL1501358 0.67 ADRA2C (0.52) CYP11B1CYP11B2CYP17A1CYP19A1SMN1; SMN2
SCHEMBL27930849 0.67 TDP1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343756-A2 1-ARYL- OR 1-ALKYLSULFONYL-HETEROCYCLYLBENZAZOLES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS Wyeth (US) 2003-09-17 EP disclosed
WO-2002036562-A2 1-ARYL- OR 1-ALKYLSULFONYL-HETEROCYCLYLBENZAZOLES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS WYETH (US) 2002-05-10 WO disclosed