SCHEMBL6972772

SCHEMBL6972772

CC(C)c1nc(CNC(N)=O)n(Cc2cccnc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.44
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CACNA1I Q9P0X4 1/20 0.38
ALDH1A1 P00352 4/20 0.38
MAPT P10636 2/20 0.38
HPGD P15428 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
S1PR3 Q99500 3/20 0.38
NAMPT P43490 2/20 0.38
ADRA1D P25100 1/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085900 0.93 ALDH1A1 (0.46) RECQLMEN1KMT2AALDH1A1MAPT
SCHEMBL6972982 0.92 MEN1 (0.41) MEN1KMT2ACACNA1IALDH1A1MAPT
SCHEMBL6970008 0.90 PIM1 (0.36) MEN1KMT2AALDH1A1KDM4ES1PR3
SCHEMBL6975509 0.90 RECQL (0.44) RECQLS1PR3NAMPTLMNACYP1A2
SCHEMBL8109122 0.89 RECQL (0.47) RECQLKMT2AALDH1A1HPGDS1PR3
SCHEMBL7086713 0.88 KMT2A (0.35) MEN1KMT2ACACNA1IALDH1A1MAPT
SCHEMBL6957033 0.87 ADRA1D (0.37) MEN1KMT2ACACNA1IALDH1A1S1PR3
SCHEMBL7078779 0.86 ADRA1D (0.35) MEN1KMT2ACACNA1IALDH1A1HPGD
SCHEMBL6973170 0.86 RECQL (0.43) RECQLKMT2AALDH1A1S1PR3NAMPT
SCHEMBL6973652 0.86 SRC (0.37) MEN1KMT2ACACNA1IALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed