SCHEMBL6973652

SCHEMBL6973652

CC(C)c1nc(CO)n(Cc2cccnc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.37
GABRA5 P31644 3/20 0.36
GABRA1 P14867 2/20 0.36
KMT2A Q03164 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
PKM P14618 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
CACNA1I Q9P0X4 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.33
ALOX5AP P20292 1/20 0.33
ADRA1D P25100 1/20 0.33
GRIN1 Q05586 2/20 0.33
GRIN2B Q13224 2/20 0.33
TLR7 Q9NYK1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7087528 0.92 SRC (0.35) SRCGABRA5GABRA1KMT2ATDP1
SCHEMBL6970034 0.92 ALDH1A1 (0.40) SRCGABRA5GABRA1KMT2ATDP1
SCHEMBL6969270 0.91 TLR7 (0.35) SRCGABRA5GABRA1KMT2ATDP1
SCHEMBL6957238 0.90 GABRA5 (0.36) SRCGABRA5GABRA1KMT2ATDP1
SCHEMBL6966848 0.90 TDP1 (0.42) KMT2ATDP1KDM4EMEN1MAPT
SCHEMBL6970546 0.89 SRC (0.37) SRCGABRA5GABRA1KMT2AKDM4E
SCHEMBL5852651 0.89 KCNH2 (0.35) KMT2ATDP1MEN1
SCHEMBL7078779 0.89 ADRA1D (0.35) SRCGABRA5GABRA1KMT2ATDP1
SCHEMBL7086713 0.88 KMT2A (0.35) SRCGABRA5GABRA1KMT2ATDP1
SCHEMBL6967631 0.88 CHRNB2 (0.39) SRCGABRA5GABRA1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed