SCHEMBL6972964

SCHEMBL6972964

CC(C)C(c1ccncc1)c1nc(CCCOCc2ccccc2)[nH]c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.37
HRH4 Q9H3N8 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
REN P00797 1/20 0.32
TACR1 P25103 2/20 0.31
TDP1 Q9NUW8 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5853119 0.90 TACR1 (0.34) GSK3BTACR1
SCHEMBL6971468 0.86 HRH4 (0.36) GSK3BHRH4HRH3RENTACR1
SCHEMBL6971688 0.82 GSK3B (0.31) GSK3B
SCHEMBL6971891 0.81 ALDH1A1 (0.37) GSK3BHRH4HRH3RENTACR1
SCHEMBL5852653 0.79 TDP1 (0.32) GSK3BTDP1
SCHEMBL6973234 0.79 GSK3B (0.31) GSK3B
SCHEMBL6973398 0.78
SCHEMBL6960435 0.77 HCAR2 (0.31) HRH3TACR1L3MBTL1
SCHEMBL5852656 0.77 GSK3B (0.32) GSK3B
SCHEMBL5853041 0.76 GSK3B (0.31) GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed