SCHEMBL6971468

SCHEMBL6971468

CC(C)c1nc(CCCOCc2ccccc2)[nH]c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
TDP1 Q9NUW8 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GSK3B P49841 2/20 0.33
REN P00797 7/20 0.32
TACR1 P25103 2/20 0.32
CAPN1 P07384 1/20 0.32
SOAT1 P35610 1/20 0.31
TUBB4A P04350 1/20 0.30
TUBB P07437 1/20 0.30
TUBA3C P0DPH7 1/20 0.30
TUBA1B P68363 1/20 0.30
TUBA4A P68366 1/20 0.30
TUBB4B P68371 1/20 0.30
TUBB3 Q13509 1/20 0.30
TUBB2A Q13885 1/20 0.30
TUBB8 Q3ZCM7 1/20 0.30
TUBA3E Q6PEY2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971891 0.94 ALDH1A1 (0.37) HRH4HRH3TDP1L3MBTL1ALDH1A1
SCHEMBL5852619 0.89 TACR1 (0.34) TDP1L3MBTL1TACR1CAPN1
SCHEMBL6972964 0.86 GSK3B (0.37) HRH4HRH3TDP1L3MBTL1GSK3B
SCHEMBL14001863 0.81 HSP90B1 (0.31)
SCHEMBL6964698 0.81 LMNA (0.36) TDP1TACR1
SCHEMBL6962307 0.78 CYP1A2 (0.35) TDP1ALDH1A1REN
SCHEMBL6975492 0.77 HRH4 (0.35) HRH4HRH3TDP1L3MBTL1GSK3B
SCHEMBL14439826 0.77 TSHR (0.39) ALDH1A1CAPN1
SCHEMBL6962088 0.76 HRH4 (0.43) HRH4HRH3TDP1L3MBTL1ALDH1A1
SCHEMBL6974600 0.76 TSHR (0.33) ALDH1A1TACR1CAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed