SCHEMBL6973071

SCHEMBL6973071

Cc1cc(C2CCN(S(=O)(=O)C3(C(=O)O)CCN(Cc4ccccc4)C(C)C3)CC2)ccc1Br

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
SIGMAR1 Q99720 5/20 0.35
BACE1 P56817 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
MMP3 P08254 5/20 0.34
USP5 P45974 2/20 0.33
MMP2 P08253 3/20 0.33
HDAC6 Q9UBN7 1/20 0.33
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLB P06746 1/20 0.33
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
MMP14 P50281 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969295 0.87 DRD2 (0.48) DRD2MEN1KMT2ACYP3A4CYP2D6
SCHEMBL6435679 0.81 CYP3A4 (0.46) DRD2MEN1KMT2ACYP3A4CYP2D6
SCHEMBL6966717 0.79 MAPT (0.36) KMT2AMMP3USP5MMP2HDAC6
SCHEMBL6966720 0.79 MAPT (0.36) KMT2AMMP3USP5MMP2HDAC6
SCHEMBL6966714 0.79 MAPT (0.36) KMT2AMMP3USP5MMP2HDAC6
SCHEMBL6971129 0.78 MMP2 (0.48) DRD2MMP3MMP2MMP1MMP9
SCHEMBL7204028 0.77 MAPT (0.38) KMT2AMMP3USP5MMP2HDAC6
SCHEMBL7202506 0.75 MAPT (0.35) KMT2AMMP3USP5MMP2MMP1
SCHEMBL6963988 0.75 MAPT (0.35) KMT2AMMP3USP5MMP2MMP1
SCHEMBL6971622 0.75 MAPT (0.35) KMT2AMMP3USP5MMP2MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1181017-B1 METALLOPROTEASE INHIBITORS PFIZER LTD (GB) 2003-04-16 EP claimed