SCHEMBL6973525

SCHEMBL6973525

CNC(=S)OCc1nc(C(C)C)c(Sc2cccc(Cl)c2)n1Cc1ccccn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.35
MAPT P10636 2/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 4/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
PPP1CA P62136 1/20 0.33
KMT2A Q03164 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 2/20 0.33
GRM5 P41594 1/20 0.32
AGTR1 P30556 1/20 0.32
HPGD P15428 1/20 0.31
KDM4E B2RXH2 1/20 0.31
PKM P14618 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7077736 0.93 ALDH1A1 (0.33) RAB9AMAPTNPC1ALDH1A1KMT2A
SCHEMBL7182670 0.91 TLR7 (0.31) RAB9ANPC1ALDH1A1LMNATP53
SCHEMBL7082819 0.90 NPC1 (0.43) RAB9AMAPTNPC1ALDH1A1GRIN1
SCHEMBL6974025 0.90 S1PR3 (0.36) RAB9AMAPTALDH1A1GRIN1GRIN2B
SCHEMBL7081153 0.87 MAPT (0.39) RAB9AMAPTNPC1ALDH1A1CYP1A2
SCHEMBL6961267 0.87 ALDH1A1 (0.34) MAPTALDH1A1LMNATP53L3MBTL1
SCHEMBL7087594 0.87 CFTR (0.39) RAB9AMAPTNPC1ALDH1A1CYP1A2
SCHEMBL7082232 0.87 S1PR3 (0.36) P2RX3
SCHEMBL7081501 0.87 NPC1 (0.38) RAB9AMAPTNPC1ALDH1A1GRIN1
SCHEMBL6958244 0.86 TP53 (0.34) RAB9AKMT2ATP53GRM5L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed