SCHEMBL6974025

SCHEMBL6974025

CNC(=S)OCc1nc(C(C)C)c(Sc2cccc(F)c2)n1Cc1ccccn1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 8/20 0.36
GRIN1 Q05586 5/20 0.34
GRIN2B Q13224 5/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
FFAR1 O14842 1/20 0.31
ENPP2 Q13822 1/20 0.31
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7082232 0.93 S1PR3 (0.36) S1PR3ENPP2
SCHEMBL7182670 0.91 TLR7 (0.31) ALDH1A1RAB9ASMN1; SMN2
SCHEMBL6973525 0.90 RAB9A (0.35) GRIN1GRIN2BALDH1A1MAPTHPGD
SCHEMBL7081110 0.90 S1PR3 (0.39) S1PR3GRIN1GRIN2BMAPTRAB9A
SCHEMBL7084823 0.87 S1PR3 (0.39) S1PR3GRIN1GRIN2BENPP2KMT2A
SCHEMBL7087594 0.87 CFTR (0.39) S1PR3ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL7077736 0.87 ALDH1A1 (0.33) ALDH1A1MAPTHPGDRAB9ASMN1; SMN2
SCHEMBL6967842 0.87 ENPP2 (0.33) GRIN1GRIN2BENPP2
SCHEMBL7078713 0.87 S1PR3 (0.39) S1PR3GRIN1GRIN2BRAB9AENPP2
SCHEMBL6969443 0.86 DHODH (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed