SCHEMBL6973823

SCHEMBL6973823

CC(C)c1nc(CCN)n(Cc2cccnc2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 7/20 0.38
GRIN2B Q13224 7/20 0.38
CHRNA7 P36544 1/20 0.37
TLR7 Q9NYK1 4/20 0.35
IDO1 P14902 1/20 0.34
ALDH1A1 P00352 2/20 0.33
POLB P06746 1/20 0.33
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP2A6 P11509 1/20 0.33
SRC P12931 1/20 0.33
S1PR3 Q99500 1/20 0.33
GNRHR P30968 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972991 0.93 GRIN1 (0.38) GRIN1GRIN2BCHRNA7TLR7
SCHEMBL7084611 0.92 GRIN1 (0.39) GRIN1GRIN2BTLR7IDO1ALDH1A1
SCHEMBL6975018 0.90 GRIN1 (0.38) GRIN1GRIN2BTLR7IDO1SRC
SCHEMBL7086853 0.89 GRIN1 (0.37) GRIN1GRIN2BTLR7IDO1ALDH1A1
SCHEMBL7082568 0.89 CHRNA7 (0.37) GRIN1GRIN2BCHRNA7TLR7TDP1
SCHEMBL6969539 0.88 GRIN1 (0.39) GRIN1GRIN2BTLR7IDO1SRC
SCHEMBL6974036 0.88 ENPP2 (0.33) TLR7
SCHEMBL7087890 0.88 TLR7 (0.41) CHRNA7TLR7ALDH1A1CYP2A6SRC
SCHEMBL6973501 0.87 LMNA (0.40) GRIN1GRIN2BPKM
SCHEMBL7081093 0.87 GRIN1 (0.37) GRIN1GRIN2BTLR7IDO1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed