SCHEMBL6973501

SCHEMBL6973501

CC(C)c1nc(CCC(=O)O)n(Cc2cccnc2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.40
HDAC6 Q9UBN7 1/20 0.40
TBXAS1 P24557 10/20 0.38
ENPP2 Q13822 3/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
TBXA2R P21731 1/20 0.38
PKM P14618 1/20 0.37
RXFP1 Q9HBX9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8344845 0.93 PKM (0.41) LMNAHDAC6TBXAS1ENPP2GRIN1
SCHEMBL8342977 0.90 LMNA (0.45) LMNAHDAC6TBXAS1ENPP2RXFP1
SCHEMBL6969096 0.89 LMNA (0.42) LMNAHDAC6TBXAS1ENPP2TBXA2R
SCHEMBL8343038 0.89 TBXA2R (0.42) LMNAENPP2TBXA2RRXFP1
SCHEMBL6975018 0.89 GRIN1 (0.38) ENPP2GRIN1GRIN2BTBXA2RPKM
SCHEMBL7086853 0.87 GRIN1 (0.37) ENPP2GRIN1GRIN2BPKM
SCHEMBL6973823 0.87 GRIN1 (0.38) GRIN1GRIN2BPKM
SCHEMBL6972580 0.87 GRIN1 (0.36) ENPP2GRIN1GRIN2BPKM
SCHEMBL6969539 0.87 GRIN1 (0.39) GRIN1GRIN2B
SCHEMBL6974966 0.86 GRIN1 (0.36) ENPP2GRIN1GRIN2BPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed