SCHEMBL6973863

SCHEMBL6973863

CC(=O)OC(Cc1ccncc1)c1nc(Sc2cc(Cl)cc(Cl)c2)c(C(C)C)[nH]1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.32
CDK5 Q00535 3/20 0.32
CDK5R1 Q15078 3/20 0.32
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
GSK3B P49841 1/20 0.30
CYP19A1 P11511 1/20 0.30
ROCK1 Q13464 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6957342 0.92 CSNK2A2 (0.38) MEN1MAPTKMT2AKDM4EALDH1A1
SCHEMBL6972752 0.89 CDC7 (0.32) CDC7CDK5CDK5R1GSK3BCYP19A1
SCHEMBL7079125 0.87 ALDH1A1 (0.36) CDC7CDK5CDK5R1KMT2AALDH1A1
SCHEMBL6961409 0.86 DHFR (0.30)
SCHEMBL6974065 0.86
SCHEMBL6968179 0.85 CYP1A2 (0.33) CDC7GSK3B
SCHEMBL7080940 0.85 MEN1 (0.31) MEN1MAPTKMT2AKDM4EALDH1A1
SCHEMBL7078284 0.84 ROCK1 (0.33) CDC7CDK5CDK5R1ROCK1
SCHEMBL6961646 0.81 TYMS (0.31) LMNA
SCHEMBL7086368 0.81 PDE4D (0.36) CDC7MEN1MAPTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed