SCHEMBL6973913

SCHEMBL6973913

CC(C)c1nc(CC#N)n(Cc2cccnc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.36
GABRA5 P31644 3/20 0.34
GABRA1 P14867 2/20 0.34
CASP1 P29466 3/20 0.33
HSD17B10 Q99714 3/20 0.33
CASP7 P55210 2/20 0.33
KDM4E B2RXH2 2/20 0.33
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
PKM P14618 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
SRC P12931 1/20 0.33
HIF1A Q16665 1/20 0.32
ALOX5AP P20292 1/20 0.32
GRIN1 Q05586 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974920 0.93 ALDH1A1 (0.37) ARGABRA5GABRA1CASP1HSD17B10
SCHEMBL6974439 0.89 KCNH2 (0.33) TDP1
SCHEMBL6974242 0.89 GRIN1 (0.38) ARCASP1HSD17B10CASP7KDM4E
SCHEMBL6969627 0.88 RECQL (0.39) ARCASP1HSD17B10CASP7KDM4E
SCHEMBL7086713 0.88 KMT2A (0.35) GABRA5GABRA1HSD17B10KDM4EKMT2A
SCHEMBL6957238 0.87 GABRA5 (0.36) GABRA5GABRA1KMT2AALDH1A1PKM
SCHEMBL6973652 0.87 SRC (0.37) GABRA5GABRA1KDM4EKMT2AALDH1A1
SCHEMBL7087528 0.86 SRC (0.35) GABRA5GABRA1KMT2AALDH1A1PKM
SCHEMBL6967631 0.86 CHRNB2 (0.39) GABRA5GABRA1KMT2APKMOPRM1
SCHEMBL7082568 0.86 CHRNA7 (0.37) GABRA5GABRA1KMT2APKMOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed