SCHEMBL6972343

SCHEMBL6972343

CC(=O)OC(Cc1cccnc1)c1nc(C(C)C)c(Sc2cccc(F)c2)[nH]1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.36
LMNA P02545 1/20 0.35
PKM P14618 1/20 0.34
KMT2A Q03164 2/20 0.33
PTAFR P25105 2/20 0.33
GRM2 Q14416 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
GFER P55789 1/20 0.33
NAMPT P43490 1/20 0.33
KDM4E B2RXH2 1/20 0.32
HSD17B10 Q99714 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
TBXAS1 P24557 1/20 0.31
RORC P51449 1/20 0.31
SGMS2 Q8NHU3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7079754 0.93 IDO1 (0.37) IDO1KMT2AGRM2NAMPTKDM4E
SCHEMBL6973954 0.90 ROCK1 (0.32) LMNAGRM2ALDH1A1MAPT
SCHEMBL6960778 0.90 LMNA (0.34) IDO1LMNAPKMKMT2APTAFR
SCHEMBL6967430 0.90 ALDH1A1 (0.41) IDO1LMNAKMT2AALDH1A1KDM4E
SCHEMBL6969311 0.89 LMNA (0.37) IDO1LMNAKMT2ANAMPTKDM4E
SCHEMBL6962106 0.87 TP53 (0.32) IDO1LMNAKMT2AGRM2ALDH1A1
SCHEMBL6972999 0.87 RXFP1 (0.37) LMNAKMT2AALDH1A1MAPTKDM4E
SCHEMBL7083467 0.86 IDO1 (0.35) IDO1LMNAPKMKMT2APTAFR
SCHEMBL6973278 0.86 MEN1 (0.35) IDO1LMNAKMT2AALDH1A1NAMPT
SCHEMBL6974498 0.85 SLC6A9 (0.35) LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed