SCHEMBL6974042

SCHEMBL6974042

CCn1c(C=O)nc(C(C)C)c1Sc1cccc(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
TERT O14746 1/20 0.36
TDP1 Q9NUW8 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TYMS P04818 2/20 0.34
VDR P11473 1/20 0.34
DHFR P00374 1/20 0.33
PTGER4 P35408 1/20 0.33
POLB P06746 1/20 0.33
ALOX12 P18054 1/20 0.33
GRM5 P41594 2/20 0.33
AKR1B1 P15121 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969836 0.88 HSP90B1 (0.32) PTGER4
SCHEMBL6968637 0.86 DHODH (0.34) KMT2ATYMSDHFRPTGER4LMNA
SCHEMBL6969927 0.86 IDO1 (0.38) TP53RXFP1TERTTDP1MEN1
SCHEMBL6973443 0.86 TP53 (0.35) TP53RXFP1TDP1MEN1KMT2A
SCHEMBL6973441 0.86 TP53 (0.35) TP53RXFP1TDP1MEN1KMT2A
SCHEMBL6969032 0.86 KDM4E (0.33) NPSR1L3MBTL1VDRPTGER4POLB
SCHEMBL6967902 0.85 NPSR1 (0.39) TP53RXFP1TERTTDP1MEN1
SCHEMBL6973903 0.84 GRIN1 (0.38) TP53RXFP1TDP1MEN1KMT2A
SCHEMBL6970594 0.83 ALDH1A1 (0.40) TP53TDP1KMT2ALMNA
SCHEMBL6973701 0.83 SMN1; SMN2 (0.40) MEN1KMT2ANPSR1L3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed