SCHEMBL6974995

SCHEMBL6974995

CC(C)c1nc(CCCO)n(Cc2ccccn2)c1Sc1cccc(F)c1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 8/20 0.36
GRIN2B Q13224 8/20 0.36
TLR7 Q9NYK1 1/20 0.34
S1PR3 Q99500 2/20 0.34
GCGR P47871 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HRH1 P35367 1/20 0.32
TSHR P16473 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
KMT2A Q03164 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973313 0.94 GRIN1 (0.38) GRIN1GRIN2BTLR7S1PR3GCGR
SCHEMBL6973869 0.93 TLR7 (0.35) GRIN1GRIN2BTLR7S1PR3KDM4E
SCHEMBL6967980 0.91 GRIN1 (0.39) GRIN1GRIN2BS1PR3GCGRKDM4E
SCHEMBL7084830 0.90 TLR7 (0.40) TLR7HRH1TSHRKMT2AALDH1A1
SCHEMBL6974023 0.89 TLR8 (0.36) GRIN1GRIN2BTLR7KDM4EHRH1
SCHEMBL6974115 0.89 GRIN1 (0.38) GRIN1GRIN2BTLR7S1PR3KDM4E
SCHEMBL6974453 0.88 ENPP2 (0.38) GRIN1GRIN2BS1PR3KMT2A
SCHEMBL6972948 0.87 GRIN1 (0.39) GRIN1GRIN2BTLR7S1PR3KDM4E
SCHEMBL6967358 0.87 S1PR3 (0.35) GRIN1GRIN2BTLR7S1PR3KDM4E
SCHEMBL6974365 0.87 GRIN1 (0.35) GRIN1GRIN2BS1PR3HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed