SCHEMBL7078281

SCHEMBL7078281

CC(=O)OCc1nc(Sc2cccc(F)c2)c(C(C)C)n1Cc1ccncc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.36
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
S1PR3 Q99500 2/20 0.33
CYP3A4 P08684 3/20 0.33
CYP2D6 P10635 3/20 0.33
CYP2C9 P11712 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C19 P33261 2/20 0.33
USP2 O75604 2/20 0.33
MIF P14174 1/20 0.33
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
MAPT P10636 1/20 0.32
SLC6A9 P48067 2/20 0.32
CA2 P00918 1/20 0.32
CA4 P22748 1/20 0.32
GRM2 Q14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7081063 0.92 ENPP2 (0.35) ENPP2LMNATP53GRIN1GRIN2B
SCHEMBL6972748 0.92 ENPP2 (0.35) ENPP2LMNATP53S1PR3ALDH1A1
SCHEMBL6957340 0.90 CSNK2A2 (0.38) TP53S1PR3ALDH1A1HPGDMAPT
SCHEMBL7079123 0.89 MEN1 (0.37) ENPP2TP53S1PR3CYP2C9CYP1A2
SCHEMBL7086366 0.87 PDE4A (0.37) LMNACYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL7086265 0.87 CA2 (0.36) LMNAS1PR3CYP2C9CYP1A2CYP2C19
SCHEMBL6974317 0.86 GRIN1 (0.36) LMNATP53GRIN1GRIN2BS1PR3
SCHEMBL7086504 0.86 GRIN1 (0.33) LMNATP53GRIN1GRIN2BS1PR3
SCHEMBL6973952 0.86 ENPP2 (0.36) ENPP2LMNATP53GRIN1GRIN2B
SCHEMBL6973861 0.85 MEN1 (0.33) ENPP2LMNAS1PR3ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed