SCHEMBL6961097

SCHEMBL6961097

CC(C)c1c(Sc2cccc(F)c2)nc(CN)n1Cc1ccncc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
ATM Q13315 2/20 0.33
KMT2A Q03164 1/20 0.33
KCNK13 Q9HB14 4/20 0.32
P2RX3 P56373 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP17A1 P05093 1/20 0.32
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
S1PR3 Q99500 1/20 0.31
HTR1A P08908 1/20 0.31
DRD2 P14416 1/20 0.31
HTR2A P28223 1/20 0.31
HTR7 P34969 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7079972 0.91 KCNK13 (0.32) GRIN1GRIN2BKCNK13S1PR3
SCHEMBL6974317 0.90 GRIN1 (0.36) GRIN1GRIN2BLMNATP53ATM
SCHEMBL7085126 0.89 ALDH1A1 (0.39) LMNAKMT2ACYP11B1CYP11B2CYP3A4
SCHEMBL6973201 0.87 KDM4E (0.36) KCNK13CYP3A4S1PR3HTR6KDM4E
SCHEMBL7081063 0.85 ENPP2 (0.35) GRIN1GRIN2BLMNATP53L3MBTL1
SCHEMBL7083636 0.85 CA2 (0.36) ATMKMT2AL3MBTL1CA2CA4
SCHEMBL7078281 0.84 ENPP2 (0.36) GRIN1GRIN2BLMNATP53CYP3A4
SCHEMBL7086504 0.84 GRIN1 (0.33) GRIN1GRIN2BLMNATP53ATM
SCHEMBL6971599 0.84 GRIN1 (0.36) GRIN1GRIN2BLMNATP53ATM
SCHEMBL7077096 0.84 PDE4A (0.39) LMNAKMT2AL3MBTL1CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed