SCHEMBL6974486

SCHEMBL6974486

CC(C)c1nc(CCCO)n(Cc2ccc(N)cc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 6/20 0.35
HSP90B1 P14625 2/20 0.35
TRAP1 Q12931 2/20 0.35
ALDH1A1 P00352 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
TLR7 Q9NYK1 4/20 0.34
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6961597 0.94 HSP90B1 (0.32) TLR8HSP90B1TRAP1ALDH1A1TDP1
SCHEMBL7078876 0.91 TLR7 (0.38) TLR8HSP90B1TRAP1ALDH1A1TDP1
SCHEMBL6971451 0.90 HSP90B1 (0.33) HSP90B1TRAP1ALDH1A1TDP1HSP90AA1
SCHEMBL7083336 0.89 ALDH1A1 (0.34) ALDH1A1TDP1TLR7
SCHEMBL6966489 0.89 TLR8 (0.35) TLR8HSP90B1TRAP1ALDH1A1TDP1
SCHEMBL6962112 0.86 PPARG (0.34) TLR8TLR7
SCHEMBL8111521 0.86 P2RX3 (0.37) ALDH1A1TDP1TLR7
SCHEMBL6968855 0.85 ALDH1A1 (0.36) TLR8HSP90B1TRAP1ALDH1A1TDP1
SCHEMBL6961149 0.85 P2RX3 (0.35) TLR8ALDH1A1TDP1
SCHEMBL6969270 0.85 TLR7 (0.35) TLR8ALDH1A1TDP1TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed