SCHEMBL6974725

SCHEMBL6974725

CC(C)c1nc(CNC(N)=O)n(Cc2ccncc2)c1Sc1cccc(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.37
LMNA P02545 3/20 0.37
ALDH1A1 P00352 2/20 0.37
TP53 P04637 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PIM1 P11309 1/20 0.36
PIM3 Q86V86 1/20 0.36
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
IDO1 P14902 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
CSNK2A2 P19784 1/20 0.34
CSNK2B P67870 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
NAMPT P43490 1/20 0.34
FLT1 P17948 1/20 0.34
KDR P35968 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974067 0.92 POLB (0.38) POLBLMNAALDH1A1TP53NPSR1
SCHEMBL6970008 0.92 PIM1 (0.36) POLBLMNAALDH1A1TP53PIM1
SCHEMBL7085900 0.91 ALDH1A1 (0.46) POLBLMNAALDH1A1TP53NPSR1
SCHEMBL7087801 0.90 ROCK2 (0.36) LMNATP53PIM1PIM3ROCK2
SCHEMBL6961674 0.90 TP53 (0.39) LMNAALDH1A1TP53PIM1PIM3
SCHEMBL6972144 0.88 IDO1 (0.35) POLBLMNAALDH1A1TP53NPSR1
SCHEMBL6972417 0.88 TP53 (0.39) POLBLMNAALDH1A1TP53HTT
SCHEMBL7086267 0.87 MAPT (0.42) POLBLMNAALDH1A1TP53
SCHEMBL7085418 0.87 POLB (0.38) POLBALDH1A1TP53RXFP1S1PR3
SCHEMBL6960281 0.86 PIM1 (0.36) POLBTP53PIM1PIM3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed