SCHEMBL6972417

SCHEMBL6972417

CCn1c(CNC(N)=O)nc(C(C)C)c1Sc1cccc(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.39
RXFP1 Q9HBX9 1/20 0.39
POLB P06746 1/20 0.36
TYMS P04818 1/20 0.35
CNR2 P34972 1/20 0.35
LMNA P02545 2/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HTT P42858 1/20 0.34
AKR1B1 P15121 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
ALOX12 P18054 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6975217 0.91 TP53 (0.39) TP53RXFP1POLBCNR2LMNA
SCHEMBL6974137 0.90 CYP2C9 (0.32) LMNAHTT
SCHEMBL6968447 0.88 CA2 (0.38) TYMSLMNAHTTALDH1A1
SCHEMBL6971356 0.88 TP53 (0.38) TP53RXFP1POLBTYMSLMNA
SCHEMBL6974725 0.88 POLB (0.37) TP53RXFP1POLBLMNAHTT
SCHEMBL7086092 0.87 LMNA (0.35) TP53POLBLMNAMEN1KMT2A
SCHEMBL7080431 0.86 MEN1 (0.36) TP53RXFP1POLBTYMSLMNA
SCHEMBL7085418 0.85 POLB (0.38) TP53RXFP1POLBKMT2AALDH1A1
SCHEMBL6972949 0.85 ALOX12 (0.37) TP53RXFP1TYMSSMN1; SMN2AKR1B1
SCHEMBL7085900 0.85 ALDH1A1 (0.46) TP53POLBLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed