SCHEMBL6961674

SCHEMBL6961674

CC(C)c1nc(CNC(N)=O)n(Cc2ccncc2)c1Sc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.39
ALDH1A1 P00352 4/20 0.38
CYP3A4 P08684 1/20 0.38
PIM1 P11309 1/20 0.37
PIM3 Q86V86 1/20 0.37
KLKB1 P03952 1/20 0.36
S1PR3 Q99500 1/20 0.36
EGLN1 Q9GZT9 1/20 0.35
GAA P10253 2/20 0.35
RECQL P46063 1/20 0.34
MAPT P10636 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
BRD4 O60885 1/20 0.34
TRPA1 O75762 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7082255 0.91 ALDH1A1 (0.41) TP53ALDH1A1CYP3A4KLKB1S1PR3
SCHEMBL6974725 0.90 POLB (0.37) TP53ALDH1A1PIM1PIM3S1PR3
SCHEMBL8109122 0.89 RECQL (0.47) TP53ALDH1A1CYP3A4S1PR3RECQL
SCHEMBL7087801 0.89 ROCK2 (0.36) TP53CYP3A4PIM1PIM3S1PR3
SCHEMBL6970008 0.88 PIM1 (0.36) TP53ALDH1A1PIM1PIM3S1PR3
SCHEMBL6974781 0.87 ENPP2 (0.35) TP53PIM1PIM3S1PR3MAPT
SCHEMBL6960328 0.86 ALDH1A1 (0.37) TP53ALDH1A1CYP3A4KLKB1MAPT
SCHEMBL7086267 0.86 MAPT (0.42) TP53ALDH1A1RECQLMAPTMEN1
SCHEMBL7086092 0.85 LMNA (0.35) TP53ALDH1A1RECQLMAPTSMN1; SMN2
SCHEMBL6972373 0.85 PIM1 (0.36) TP53ALDH1A1PIM1PIM3GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed