SCHEMBL6975989

SCHEMBL6975989

Cn1c(CO)cnc1Cc1ccc(Cl)cc1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.59
NPC1 O15118 1/20 0.59
RECQL P46063 1/20 0.57
ALDH1A1 P00352 3/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48
HRH3 Q9Y5N1 2/20 0.45
KMT2A Q03164 5/20 0.42
MEN1 O00255 3/20 0.42
MAPK1 P28482 1/20 0.40
KDM4E B2RXH2 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
NOTUM Q6P988 1/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14028404 0.75 RAB9A (1.00) RAB9ANPC1RECQLALDH1A1LMNA
SCHEMBL10288448 0.72 CYP2C19 (0.44) RAB9ANPC1RECQLALDH1A1LMNA
SCHEMBL6969631 0.70 HSD11B1 (0.44) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL13059104 0.70
SCHEMBL6778626 0.68 ALDH1A1 (0.40) RAB9ANPC1RECQLALDH1A1LMNA
SCHEMBL14012156 0.68 ALDH1A1 (0.40) RAB9ANPC1RECQLALDH1A1LMNA
SCHEMBL8126668 0.68 MAPK1 (0.54) RAB9ANPC1RECQLALDH1A1LMNA
SCHEMBL27553901 0.67 ALDH1A1 (0.39) RAB9ANPC1ALDH1A1KMT2AMEN1
SCHEMBL14037790 0.65 CYP2C19 (0.38) RAB9ANPC1RECQLALDH1A1LMNA
SCHEMBL8992959 0.65 IDO1 (0.46) ALDH1A1LMNAMAPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6566376-B1 For therapy of chemokine receptor related diseases and conditions such as rheumatoid arthritis, chronic obstructive pulmonary disease ASTRAZENECA UK LIMITED (GB) 2003-05-20 US disclosed
EP-1202984-B1 DIPHENYL-PIPERIDINE DERIVATE ASTRAZENECA UK LTD (GB) 2003-03-05 EP disclosed