SCHEMBL6976473

SCHEMBL6976473

N=C(N)NCCC[C@@H](C(=O)c1nc2ccc(C(=O)O)cc2s1)N1CCC[C@H]1C(N)=O

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.37
NPC1 O15118 8/20 0.37
NFKB1 P19838 2/20 0.37
NFKB2 Q00653 2/20 0.37
RELA Q04206 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MITF O75030 1/20 0.37
TP53 P04637 1/20 0.37
PKM P14618 1/20 0.37
LMNA P02545 1/20 0.35
F2 P00734 2/20 0.35
TMPRSS15 P98073 1/20 0.35
MAOB P27338 3/20 0.35
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
DPP4 P27487 2/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976769 0.91 MAOB (0.44) MAOBDPP4
SCHEMBL6976617 0.90 SMYD3 (0.42) RAB9ANPC1SMN1; SMN2TP53LMNA
SCHEMBL6976833 0.89 F2 (0.36) RAB9ANPC1TP53F2MAOB
SCHEMBL6976541 0.88 MAOB (0.47) RAB9ANPC1NFKB1NFKB2RELA
SCHEMBL6972547 0.88 F2 (0.43) F2MAOB
SCHEMBL6975942 0.88 F2 (0.35) RAB9ANPC1NFKB1NFKB2RELA
SCHEMBL6976859 0.84 F2 (0.39) SMN1; SMN2F2
SCHEMBL17145025 0.81 NFKB1 (0.41) RAB9ANPC1NFKB1NFKB2RELA
SCHEMBL17145027 0.81 NFKB1 (0.41) RAB9ANPC1NFKB1NFKB2RELA
SCHEMBL6972814 0.79 DPP4 (0.34) LMNADPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0833839-B1 PEPTIDYL HETEROCYCLES USEFUL IN THE TREATMENT OF THROMBIN RELATED DISORDERS ORTHO PHARMA CORP (US) 2003-01-08 EP claimed