SCHEMBL6976685

SCHEMBL6976685

Cc1c(C)c2c(c(C)c1N)CC(C)(CN1CCC(c3cn(-c4ccccc4)c4ccccc34)CC1)O2

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.38
HTR6 P50406 4/20 0.34
HRH2 P25021 1/20 0.31
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL6983587 0.96 KCNH2 (0.37) KCNH2HTR6HRH2
SCHEMBL6981562 0.81 DRD2 (0.43) SIGMAR1
SCHEMBL6981384 0.81 DRD2 (0.43) SIGMAR1
SCHEMBL7811043 0.81 DRD2 (0.43) SIGMAR1
Hydrochloric Acid SCHEMBL7811763 0.80 DRD2 (0.42) SIGMAR1
Bromide SCHEMBL7811677 0.80 DRD2 (0.42) SIGMAR1
Bromide SCHEMBL7811682 0.80 DRD2 (0.42) SIGMAR1
Hydrochloric Acid SCHEMBL6984757 0.80 DRD2 (0.42) SIGMAR1
Hydrochloric Acid SCHEMBL6985847 0.80 DRD2 (0.42) SIGMAR1
SCHEMBL6985174 0.79 HTR6 (0.39) KCNH2HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed
EP-0923575-A1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS Takeda Chemical Industries, Ltd. (JP) 1999-06-23 EP disclosed
WO-1998008842-A1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-03-05 WO disclosed