SCHEMBL6976935

SCHEMBL6976935

Cc1c(C)c2c(c(C)c1N)CC(C)(CN1CCC(OC/C=C/c3ccccc3)CC1)O2

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.40
SIGMAR1 Q99720 8/20 0.37
HTR2A P28223 7/20 0.37
HTR2C P28335 7/20 0.37
HTR2B P41595 7/20 0.37
TMEM97 Q5BJF2 1/20 0.35
DRD2 P14416 3/20 0.33
OPRM1 P35372 1/20 0.33
AGTR2 P50052 2/20 0.33
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976937 1.00 DPP4 (0.40) DPP4SIGMAR1HTR2AHTR2CHTR2B
SCHEMBL6980205 0.84 CARM1 (0.43) DPP4SIGMAR1TMEM97OPRM1
SCHEMBL6983930 0.80 CHRM2 (0.43) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL6981384 0.79 DRD2 (0.43) SIGMAR1DRD2
SCHEMBL7811043 0.79 DRD2 (0.43) SIGMAR1DRD2
SCHEMBL6981562 0.79 DRD2 (0.43) SIGMAR1DRD2
Hydrochloric Acid SCHEMBL6985847 0.78 DRD2 (0.42) SIGMAR1DRD2
Bromide SCHEMBL7811682 0.78 DRD2 (0.42) SIGMAR1DRD2
Bromide SCHEMBL7811677 0.78 DRD2 (0.42) SIGMAR1DRD2
Hydrochloric Acid SCHEMBL6984757 0.78 DRD2 (0.42) SIGMAR1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed