SCHEMBL7079929

SCHEMBL7079929

CC(C)c1nc(CO)n(Cc2ccccn2)c1Sc1cccc(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.38
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
KDM4E B2RXH2 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
PKM P14618 1/20 0.36
ALDH1A1 P00352 5/20 0.36
KMT2A Q03164 3/20 0.36
MAPT P10636 2/20 0.36
PPP1CA P62136 1/20 0.36
TP53 P04637 2/20 0.35
MEN1 O00255 2/20 0.34
HPGD P15428 1/20 0.34
AGTR1 P30556 1/20 0.34
NPSR1 Q6W5P4 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
RAB9A P51151 2/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7082472 0.92 ALDH1A1 (0.37) GRM5GRIN1GRIN2BKDM4EL3MBTL1
SCHEMBL6976953 0.92 ALDH1A1 (0.33) GRIN1GRIN2BKDM4EALDH1A1KMT2A
SCHEMBL6974023 0.91 TLR8 (0.36) GRM5GRIN1GRIN2BKDM4EL3MBTL1
SCHEMBL6962202 0.90 GRM5 (0.38) GRM5GRIN1GRIN2BKDM4EL3MBTL1
SCHEMBL6963974 0.89 ALDH1A1 (0.37) KDM4EL3MBTL1ALDH1A1TP53NPSR1
SCHEMBL6967528 0.89 GRM5 (0.36) GRM5GRIN1GRIN2BKDM4EL3MBTL1
SCHEMBL6961462 0.89 GRIN1 (0.37) GRM5GRIN1GRIN2BKDM4EL3MBTL1
SCHEMBL7079263 0.89 SLC6A2 (0.41) GRM5GRIN1GRIN2BKDM4EL3MBTL1
SCHEMBL6960270 0.88 ALDH1A1 (0.36) GRM5GRIN1GRIN2BKDM4EL3MBTL1
SCHEMBL6967980 0.88 GRIN1 (0.39) GRIN1GRIN2BKDM4EALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed