SCHEMBL6977874

SCHEMBL6977874

COC(=O)CC(c1ccco1)C1CCCCC(=N)N1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
POLB P06746 3/20 0.43
HPGD P15428 3/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KDM4E B2RXH2 2/20 0.35
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CYP2C19 P33261 2/20 0.33
ALOX15 P16050 1/20 0.32
ATM Q13315 1/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974191 0.80 YAP1 (0.35) TSHRSLC6A3
SCHEMBL6978293 0.79 ALDH1A1 (0.39) ALDH1A1POLBHPGDKDM4ERAB9A
SCHEMBL6977392 0.77 ALDH1A1 (0.37) ALDH1A1POLB
Trifluoroacetic Acid SCHEMBL6981240 0.77 ALDH1A1 (0.41) ALDH1A1POLBHPGDSMN1; SMN2KDM4E
SCHEMBL6966808 0.77 ALDH1A1 (0.35) ALDH1A1POLBTP53MAPTNPSR1
SCHEMBL6972056 0.77 MAPT (0.35) MAPT
SCHEMBL6976352 0.68 ALDH1A1 (0.42) ALDH1A1POLBHPGDSMN1; SMN2KDM4E
SCHEMBL6981063 0.68 ALDH1A1 (0.31) ALDH1A1POLBMAPT
SCHEMBL6978310 0.67 ALDH1A1 (0.41) ALDH1A1POLBHPGDSMN1; SMN2KDM4E
SCHEMBL5468924 0.66 KCNA5 (0.41) ALDH1A1TSHRSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883251-A ENZYME INHIBITORS G. D. SEARLE & CO. (US) 1999-03-16 US claimed
EP-0821674-B1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2003-08-06 EP disclosed
US-6011028-A Cyclic amidino agents useful as nitric oxide synthase inhibitors G.D. SEARLE & CO. (US) 2000-01-04 US disclosed
EP-0821674-A1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1998-02-04 EP disclosed