SCHEMBL6978036

SCHEMBL6978036

Nc1nc(N)nc(C2CCN(c3ccc(-c4ccccc4)cc3)CC2)n1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DHFR P00374 9/20 0.50
HRH3 Q9Y5N1 1/20 0.43
MAPT P10636 1/20 0.40
GFER P55789 1/20 0.40
ADORA2A P29274 2/20 0.40
ADORA1 P30542 2/20 0.40
POLB P06746 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
ADORA2B P29275 1/20 0.40
HTR1A P08908 1/20 0.39
DRD2 P14416 1/20 0.39
HTR2A P28223 1/20 0.39
HTR7 P34969 1/20 0.39
HTR6 P50406 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982632 0.91 DHFR (0.48) DHFRMAPTGFERHTR1ADRD2
SCHEMBL6983539 0.78 DHFR (0.51) DHFRHRH3MAPTDRD2
SCHEMBL6981484 0.72 DRD2 (0.58) HRH3POLBDRD2
SCHEMBL6982266 0.71 DHFR (0.45) DHFRMAPTADORA2AADORA1POLB
SCHEMBL6982271 0.71 DHFR (0.45) DHFRMAPTADORA2AADORA1POLB
SCHEMBL3900451 0.71 HRH3 (0.51) HRH3MAPTPOLBFFAR4
Fluoride SCHEMBL27569822 0.69 MEN1 (0.56) DHFRMAPTPOLBHTR7
Biphenyl SCHEMBL183386 0.69 ADORA2A (0.75) DHFRADORA2AADORA1POLBADORA3
SCHEMBL241159 0.68 DHFR (0.50) DHFRMAPTGFERPOLBDRD2
SCHEMBL21460347 0.68 NAMPT (0.50) HRH3FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1037886-B1 TRIAZINE ANGIOGENESIS INHIBITORS ABBOTT LAB (US) 2003-05-02 EP claimed
US-6288228-B1 DIAMINOTRIAZINE DERIVATIVES ABBOTT LABORATORIES 2001-09-11 US claimed
US-6150362-A ADMINISTERING 1,3,5-SUBSTITUTED TRIAZINE COMPOUNDS TO THE PATIENT SUFFERING FROM ANGIOGENIC DISEASES ABBVIE INC. 2000-11-21 US claimed
EP-1037886-B1 TRIAZINE ANGIOGENESIS INHIBITORS ABBOTT LAB (US) 2003-05-02 EP disclosed
US-6288228-B1 DIAMINOTRIAZINE DERIVATIVES ABBOTT LABORATORIES 2001-09-11 US disclosed
US-6150362-A ADMINISTERING 1,3,5-SUBSTITUTED TRIAZINE COMPOUNDS TO THE PATIENT SUFFERING FROM ANGIOGENIC DISEASES ABBVIE INC. 2000-11-21 US disclosed
EP-1037886-A1 TRIAZINE ANGIOGENESIS INHIBITORS Abbott Laboratories (US) 2000-09-27 EP disclosed
WO-1999031088-A1 TRIAZINE ANGIOGENESIS INHIBITORS ABBOTT LABORATORIES (US) 1999-06-24 WO disclosed