SCHEMBL6978239

SCHEMBL6978239

Cc1c(C)c2c(c(C)c1N)CC(C)(CN1CCC(NC(c3ccc(F)cc3)c3ccc(F)cc3)CC1)O2

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 7/20 0.37
CHRM1 P11229 6/20 0.37
SLC6A2 P23975 6/20 0.37
SLC6A3 Q01959 4/20 0.36
KCNH2 Q12809 1/20 0.34
OPRM1 P35372 1/20 0.32
DRD2 P14416 1/20 0.30
DRD4 P21917 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980124 0.91 CHRM1 (0.32) SLC6A4CHRM1SLC6A2
SCHEMBL6976347 0.91 CHRM1 (0.32) SLC6A4CHRM1SLC6A2
SCHEMBL6983686 0.91 CHRM1 (0.32) SLC6A4CHRM1SLC6A2
Hydrochloric Acid SCHEMBL6980788 0.90 CHRM1 (0.31) SLC6A4CHRM1SLC6A2
SCHEMBL6984267 0.89 CXCR3 (0.31)
Sulfuric Acid SCHEMBL6984280 0.86 MGLL (0.31)
Sulfuric Acid SCHEMBL6985648 0.86 MGLL (0.31)
Sulfuric Acid SCHEMBL6984275 0.86 MGLL (0.31)
SCHEMBL6977637 0.83 CHRM1 (0.30) SLC6A4CHRM1SLC6A2
Oxalic Acid SCHEMBL6985362 0.79 BCHE (0.40) SLC6A4SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed