SCHEMBL6979842

SCHEMBL6979842

N=C(N)c1ccc(NC(=O)CCC(=O)NCC(C(=O)O)c2ncc[nH]2)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 1/20 0.38
KLK1 P06870 2/20 0.37
KLK5 Q9Y337 2/20 0.37
ITGB3 P05106 3/20 0.36
ITGA2B P08514 3/20 0.36
F10 P00742 8/20 0.36
F9 P00740 4/20 0.35
PRSS1 P07477 2/20 0.35
F2 P00734 2/20 0.35
TMPRSS15 P98073 1/20 0.35
PLAU P00749 1/20 0.35
HPN P05981 1/20 0.35
F7 P08709 3/20 0.34
KLKB1 P03952 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982101 0.90 F7 (0.39) FPR2KLK1KLK5ITGB3ITGA2B
SCHEMBL6982365 0.80 ALDH1A1 (0.34)
SCHEMBL6980170 0.80 KLK1 (0.39) KLK1KLK5ITGB3ITGA2BF10
SCHEMBL6976581 0.74 ITGB3 (0.48) KLK1KLK5ITGB3ITGA2BF7
SCHEMBL6982666 0.73 ADORA2A (0.41) KLK1KLK5ITGB3ITGA2BF10
SCHEMBL9262501 0.72 KLK1 (0.42) FPR2KLK1KLK5ITGB3ITGA2B
SCHEMBL6985138 0.71 ITGB3 (0.36) ITGB3ITGA2BPRSS1TMPRSS15
SCHEMBL9263614 0.70 KLK5 (0.40) KLK1KLK5ITGB3ITGA2BF10
SCHEMBL6985761 0.70 BRD4 (0.37) F7
SCHEMBL6983774 0.69 ADORA2A (0.40) ITGB3ITGA2BF10PRSS1F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630366-B1 SUBSTITUTED HETEROCYCLIC DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 2003-01-02 EP disclosed
EP-0539343-B1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO CO (US) 2000-07-26 EP disclosed
US-5378727-A ADMINISTERING TO MAMMALS G. D. SEARLE & CO. (US) 1995-01-03 US disclosed
US-5254573-A Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-10-19 US disclosed
EP-0539343-A1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-04-28 EP disclosed