SCHEMBL6983774

SCHEMBL6983774

N=C(N)c1cc(F)c(NC(=O)CCC(=O)NCC(C(=O)O)c2nccs2)c(F)c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.40
ADORA1 P30542 2/20 0.40
ADORA2B P29275 1/20 0.40
KLKB1 P03952 1/20 0.35
HDAC3 O15379 2/20 0.34
HDAC1 Q13547 2/20 0.34
ITGB3 P05106 6/20 0.34
ITGA2B P08514 6/20 0.34
SLC6A9 P48067 1/20 0.34
F7 P08709 2/20 0.33
F2 P00734 1/20 0.33
F10 P00742 1/20 0.33
PLG P00747 1/20 0.33
F3 P13726 1/20 0.33
TMPRSS15 P98073 4/20 0.32
PRSS1 P07477 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977286 0.83 ITGB3 (0.53) ADORA2AITGB3ITGA2BF7F2
SCHEMBL6982666 0.77 ADORA2A (0.41) ADORA2AADORA1KLKB1HDAC3HDAC1
SCHEMBL6985138 0.77 ITGB3 (0.36) ITGB3ITGA2BTMPRSS15PRSS1
SCHEMBL6983709 0.75 HDAC3 (0.36) HDAC3HDAC1SLC6A9
SCHEMBL8042923 0.69 ITGB3 (0.49) ITGB3ITGA2B
SCHEMBL6979842 0.69 FPR2 (0.38) KLKB1ITGB3ITGA2BF7F2
SCHEMBL6980649 0.67 ADORA2A (0.41) ADORA2AITGB3ITGA2BF7F2
SCHEMBL6980170 0.67 KLK1 (0.39) ADORA2AADORA1HDAC3HDAC1ITGB3
SCHEMBL6984634 0.67 ITGB3 (0.46) ITGB3ITGA2BF7F2F10
SCHEMBL6982396 0.67 ITGB3 (0.35) ITGB3ITGA2BF2F10PLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630366-B1 SUBSTITUTED HETEROCYCLIC DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 2003-01-02 EP disclosed
EP-0539343-B1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO CO (US) 2000-07-26 EP disclosed
US-5378727-A ADMINISTERING TO MAMMALS G. D. SEARLE & CO. (US) 1995-01-03 US disclosed
US-5254573-A Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-10-19 US disclosed
EP-0539343-A1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-04-28 EP disclosed