SCHEMBL6982365

SCHEMBL6982365

N=C(N)c1ccc(NC(=O)CCC(=O)NCC(C(=O)O)c2ncc[nH]2)c2ccccc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
MMP2 P08253 2/20 0.34
SHMT2 P34897 1/20 0.34
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
PGGT1B P53609 1/20 0.33
RPS6KB1 P23443 2/20 0.33
CSNK1A1 P48729 1/20 0.33
TYRO3 Q06418 1/20 0.33
DYRK1B Q9Y463 1/20 0.33
NPC1 O15118 1/20 0.32
CYP1A2 P05177 2/20 0.31
CYP2C19 P33261 2/20 0.31
SLC1A2 P43004 1/20 0.31
SLC1A1 P43005 1/20 0.31
POLB P06746 2/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
APOBEC3A P31941 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985761 0.90 BRD4 (0.37) ALDH1A1CYP1A2CYP2C19POLBKDM4E
SCHEMBL6983709 0.82 HDAC3 (0.36) ALDH1A1SHMT2RPS6KB1CYP1A2CYP2C19
SCHEMBL6979842 0.80 FPR2 (0.38)
Hydrochloric Acid SCHEMBL7346044 0.73 CYP2C19 (0.51) ALDH1A1SHMT2CYP1A2CYP2C19POLB
SCHEMBL6982101 0.70 F7 (0.39)
SCHEMBL6976581 0.69 ITGB3 (0.48) MAPT
SCHEMBL9559011 0.68 ITGB3 (0.63)
SCHEMBL9262501 0.67 KLK1 (0.42)
SCHEMBL6981209 0.67 F7 (0.39) ALDH1A1NPC1MAPTHTT
SCHEMBL9263614 0.65 KLK5 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630366-B1 SUBSTITUTED HETEROCYCLIC DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 2003-01-02 EP disclosed
EP-0539343-B1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO CO (US) 2000-07-26 EP disclosed
US-5378727-A ADMINISTERING TO MAMMALS G. D. SEARLE & CO. (US) 1995-01-03 US disclosed
US-5254573-A Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-10-19 US disclosed
EP-0539343-A1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-04-28 EP disclosed