SCHEMBL6980378

SCHEMBL6980378

O=S(=O)(Nc1cccc2cccnc12)c1cccc(Cl)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC40A1 Q9NP59 13/20 1.00
GLO1 Q04760 6/20 0.72
TDP1 Q9NUW8 4/20 0.72
G6PD P11413 1/20 0.72
NFKBIA P25963 1/20 0.72
AGTR1 P30556 1/20 0.72
METAP2 P50579 1/20 0.72
METAP1 P53582 1/20 0.72
PAX8 Q06710 1/20 0.72
ATM Q13315 1/20 0.72
MEN1 O00255 3/20 0.70
KMT2A Q03164 3/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1319547 0.90 SLC40A1 (0.82) SLC40A1GLO1TDP1G6PDNFKBIA
SCHEMBL6981081 0.86 SLC40A1 (1.00) SLC40A1GLO1TDP1G6PDNFKBIA
SCHEMBL30925586 0.86 SLC40A1 (1.00) SLC40A1GLO1TDP1G6PDNFKBIA
SCHEMBL13485937 0.85 SLC40A1 (0.74) SLC40A1GLO1TDP1G6PDNFKBIA
SCHEMBL13485928 0.85 GLO1 (0.80) SLC40A1GLO1TDP1G6PDNFKBIA
SCHEMBL442367 0.84 SLC40A1 (1.00) SLC40A1GLO1TDP1G6PDNFKBIA
SCHEMBL15508515 0.84 GLO1 (0.76) SLC40A1GLO1TDP1G6PDNFKBIA
SCHEMBL6980652 0.84 TDP1 (0.76) SLC40A1GLO1TDP1G6PDNFKBIA
SCHEMBL11973852 0.84 SLC40A1 (1.00) SLC40A1GLO1TDP1G6PDNFKBIA
SCHEMBL30925492 0.84 GLO1 (0.76) SLC40A1GLO1TDP1G6PDNFKBIA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675526-B1 NOVEL SULFONAMINOQUINOLINE HEPCIDIN ANTAGONISTS VIFOR (INTERNATIONAL) AG (CH) 2017-02-01 EP disclosed
US-9102688-B2 Sulfonaminoquinoline hepcidin antagonists VIFOR (INTERNATIONAL) AG (CH) 2015-08-11 US disclosed
US-9102688-B2 Sulfonaminoquinoline hepcidin antagonists VIFOR (INTERNATIONAL) AG (CH) 2015-08-11 US disclosed
US-9102688-B2 Sulfonaminoquinoline hepcidin antagonists VIFOR (INTERNATIONAL) AG (CH) 2015-08-11 US disclosed
US-20140364424-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2014-12-11 US disclosed
US-20140364424-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2014-12-11 US disclosed
US-20140364424-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2014-12-11 US disclosed
US-20120214803-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2012-08-23 US disclosed
US-20120214803-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2012-08-23 US disclosed
US-20120214803-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2012-08-23 US disclosed
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120214803-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists HAMP, SLC40A1, FTH1 SLC40A1 2/4885GLO1 3935/4885TDP1 4862/4885
US-20140364424-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists HAMP, SLC40A1, FTH1 SLC40A1 2/4885GLO1 3935/4885TDP1 4862/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.