SCHEMBL6981028

SCHEMBL6981028

N#Cc1ccc(CCC(=O)N2CCCc3cccc(C(=O)N(Cc4ccccc4)c4ccccc4)c32)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
CHRM2 P08172 2/20 0.40
CHRM1 P11229 2/20 0.40
CHRM3 P20309 2/20 0.40
MAPKAPK2 P49137 2/20 0.39
LTB4R2 Q9NPC1 1/20 0.39
TSHR P16473 3/20 0.37
USP2 O75604 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PTGER4 P35408 1/20 0.37
MAPT P10636 2/20 0.37
MAPK1 P28482 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
KDM1A O60341 1/20 0.37
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6984361 0.91 PTGER4 (0.39) NPC1MEN1KMT2ACHRM2CHRM1
SCHEMBL6980417 0.89 PTGER4 (0.39) NPC1MEN1KMT2ATSHRUSP2
SCHEMBL6979414 0.88 LTB4R2 (0.40) NPC1MEN1KMT2ACHRM2CHRM1
SCHEMBL6983537 0.88 PTGER4 (0.38) NPC1MEN1KMT2ACHRM2CHRM1
SCHEMBL6977399 0.85 PTGER4 (0.42) NPC1MEN1KMT2ATSHRUSP2
SCHEMBL6986008 0.84 MEN1 (0.39) NPC1MEN1KMT2ACHRM2CHRM1
SCHEMBL6981025 0.83 MEN1 (0.57) NPC1MEN1KMT2ACHRM2CHRM1
SCHEMBL6986544 0.83 PTGER4 (0.39) NPC1MEN1KMT2ATSHRUSP2
SCHEMBL7407027 0.82 AR (0.39) NPC1MEN1KMT2ATSHRUSP2
SCHEMBL6986002 0.81 RXRA (0.45) NPC1MEN1KMT2ATSHRUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed