SCHEMBL6986002

SCHEMBL6986002

CN(Cc1ccccc1)c1cccc2c1N(C(=O)CCc1ccc(C#N)cc1)CCC2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.45
RXRB P28702 1/20 0.45
RXRG P48443 1/20 0.45
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 2/20 0.40
HPGD P15428 2/20 0.40
KMT2A Q03164 2/20 0.40
USP2 O75604 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TAS2R14 Q9NYV8 1/20 0.38
CYP11B2 P19099 1/20 0.38
NPC1 O15118 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
TMEM97 Q5BJF2 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6986008 0.90 MEN1 (0.39) RXRARXRBRXRGALDH1A1MEN1
SCHEMBL6987632 0.89 ALDH1A1 (0.39) ALDH1A1MEN1HPGDKMT2AUSP2
SCHEMBL6979172 0.88 KDM1A (0.41) ALDH1A1MEN1HPGDKMT2AUSP2
SCHEMBL6977636 0.88 ALDH1A1 (0.42) ALDH1A1MEN1HPGDKMT2AUSP2
SCHEMBL6981987 0.86 PTGER4 (0.38) RXRARXRBRXRGALDH1A1MEN1
SCHEMBL6981595 0.86 LTB4R2 (0.46) ALDH1A1MEN1HPGDKMT2AUSP2
SCHEMBL6984169 0.85 KDM1A (0.38) ALDH1A1NPC1SIGMAR1TMEM97MAPT
SCHEMBL6979942 0.85 TSHR (0.38) ALDH1A1MEN1HPGDKMT2AUSP2
SCHEMBL6982692 0.84 L3MBTL1 (0.38) ALDH1A1TSHRNPC1MAPTMAPK1
SCHEMBL6982667 0.84 NR3C1 (0.41) ALDH1A1MEN1HPGDKMT2AUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed