SCHEMBL6981147

SCHEMBL6981147

COc1cc(CNCCCN2CCN3CCCCC3C2)cc(OC)c1OC

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.47
MEN1 O00255 1/20 0.44
GAA P10253 1/20 0.44
KMT2A Q03164 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5845218 0.99 MEN1 (0.46) KCNH2MEN1GAAKMT2AALDH1A1
SCHEMBL6986873 0.85 SHMT2 (0.44) KCNH2
Hydrochloric Acid SCHEMBL5840949 0.84 SHMT2 (0.44) KCNH2
SCHEMBL6985106 0.82 SIGMAR1 (0.43) KCNH2
SCHEMBL5841208 0.82 SHMT2 (0.44) KCNH2
Hydrochloric Acid SCHEMBL5840340 0.81 SHMT2 (0.43)
SCHEMBL6986781 0.81 SHMT2 (0.43) KCNH2
Hydrochloric Acid SCHEMBL5841820 0.81 SIGMAR1 (0.43) KCNH2MEN1KMT2APOLB
SCHEMBL6984898 0.81 SLC29A1 (0.69) KCNH2MEN1KMT2A
Hydrochloric Acid SCHEMBL5842747 0.80 SHMT2 (0.42) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1275647-B1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-11-12 EP disclosed
EP-1275647-A1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2003-01-15 EP disclosed