SCHEMBL6986873

SCHEMBL6986873

COc1cc(NCCCN2CCN3CCCCC3C2)cc(OC)c1OC

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SHMT2 P34897 1/20 0.44
TLR9 Q9NR96 1/20 0.43
TLR7 Q9NYK1 1/20 0.43
SLC29A1 Q99808 1/20 0.43
SIGMAR1 Q99720 5/20 0.42
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
ABCB1 P08183 1/20 0.40
CHRM5 P08912 1/20 0.40
ADRA2A P08913 1/20 0.40
CHRM1 P11229 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
CHRM3 P20309 1/20 0.40
KCNH2 Q12809 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5840949 0.99 SHMT2 (0.44) SHMT2TLR9TLR7SLC29A1SIGMAR1
SCHEMBL5841208 0.97 SHMT2 (0.44) SHMT2TLR9TLR7SLC29A1SIGMAR1
SCHEMBL6986781 0.96 SHMT2 (0.43) SHMT2TLR9TLR7SLC29A1SIGMAR1
Hydrochloric Acid SCHEMBL5840340 0.96 SHMT2 (0.43) SHMT2TLR9TLR7SLC29A1SIGMAR1
Hydrochloric Acid SCHEMBL5842747 0.95 SHMT2 (0.42) SHMT2TLR9TLR7SIGMAR1KCNH2
SCHEMBL6982261 0.85 SHMT2 (0.55) SHMT2TLR9TLR7SIGMAR1
SCHEMBL6981147 0.85 KCNH2 (0.47) KCNH2
Hydrochloric Acid SCHEMBL5845218 0.84 MEN1 (0.46) KCNH2
Hydrochloric Acid SCHEMBL5841553 0.84 SHMT2 (0.54) SHMT2TLR9TLR7SIGMAR1
SCHEMBL6984898 0.83 SLC29A1 (0.69) SLC29A1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1275647-B1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-11-12 EP disclosed
EP-1275647-A1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2003-01-15 EP disclosed