SCHEMBL6981700

SCHEMBL6981700

CCOC(=O)C(Cc1ccco1)NC(=O)CCC(=O)Nc1ccc(C=NN)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.42
POLB P06746 5/20 0.42
USP2 O75604 1/20 0.42
MAPT P10636 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NPSR1 Q6W5P4 1/20 0.40
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
RAB9A P51151 1/20 0.38
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981928 0.83 RAB9A (0.45) ALDH1A1POLBMAPTNPSR1KDM4E
SCHEMBL7344701 0.80 MAPT (0.44) ALDH1A1POLBMAPTNPSR1SMN1; SMN2
SCHEMBL7473679 0.80 ITGB3 (0.47) ALDH1A1POLBMAPTNPSR1NPC1
SCHEMBL7352508 0.79 ITGB3 (0.42) ALDH1A1POLBMAPTNPSR1ITGB3
SCHEMBL6978962 0.79 POLB (0.51) ALDH1A1POLBUSP2MAPTHSD17B10
SCHEMBL4114851 0.76 CTSS (0.42) ALDH1A1POLBUSP2MAPTHSD17B10
SCHEMBL7348958 0.76 ITGB3 (0.51) ALDH1A1POLBMAPTKDM4ENPC1
SCHEMBL7349536 0.75 ITGB3 (0.48) ALDH1A1POLBMAPTNPC1SMN1; SMN2
SCHEMBL8123529 0.75 USP2 (0.35) ALDH1A1POLBUSP2MAPTHSD17B10
SCHEMBL7346612 0.75 ITGB3 (0.50) ALDH1A1POLBUSP2MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630366-B1 SUBSTITUTED HETEROCYCLIC DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 2003-01-02 EP disclosed
EP-0539343-B1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO CO (US) 2000-07-26 EP disclosed
US-5378727-A ADMINISTERING TO MAMMALS G. D. SEARLE & CO. (US) 1995-01-03 US disclosed
US-5254573-A Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-10-19 US disclosed
EP-0539343-A1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-04-28 EP disclosed