SCHEMBL7344701

SCHEMBL7344701

CCOC(=O)C(CCc1ccccc1)NC(=O)CCC(=O)Nc1ccc(C=NN)cc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.44
RAB9A P51151 1/20 0.42
ALDH1A1 P00352 4/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
LTA4H P09960 3/20 0.41
HTT P42858 1/20 0.41
POLB P06746 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
METAP2 P50579 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8895885 0.89 TSHR (0.46) MAPTRAB9AALDH1A1TSHRLTA4H
SCHEMBL7387879 0.87 KMT2A (0.48) SMN1; SMN2POLB
SCHEMBL7473679 0.82 ITGB3 (0.47) MAPTRAB9AALDH1A1TSHRSMN1; SMN2
SCHEMBL7352508 0.81 ITGB3 (0.42) MAPTALDH1A1POLBNPSR1METAP2
SCHEMBL7386056 0.80 CTSG (0.52) ALDH1A1
SCHEMBL6981928 0.80 RAB9A (0.45) MAPTRAB9AALDH1A1SMN1; SMN2HTT
SCHEMBL6981700 0.80 ALDH1A1 (0.42) MAPTRAB9AALDH1A1SMN1; SMN2POLB
SCHEMBL7353182 0.79 ITGB3 (0.51) MAPTALDH1A1SMN1; SMN2HTTPOLB
SCHEMBL7350048 0.79 ITGB3 (0.42) MAPTALDH1A1TSHR
SCHEMBL24533895 0.78 SMN1; SMN2 (0.56) MAPTALDH1A1SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5973003-A TREATMENT OF THROMBOSIS, STROKE, MYOCARDIAL INFARCTION, INFLAMMATION AND ARTERIOSCLEROSIS G. D. SEARLE & CO. (US) 1999-10-26 US disclosed
US-5344957-A Amidinoiphenyl-substituted G.D. SEARLE & CO. (US) 1994-09-06 US disclosed
US-5239113-A Anticoagulants MONSANTO COMPANY (US) 1993-08-24 US disclosed
EP-0542708-A1 Substituted B-amino acid derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-05-19 EP disclosed
WO-1993007867-A1 SUBSTITUTED β-AMINO ACID DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1993-04-29 WO disclosed