SCHEMBL6982745

SCHEMBL6982745

CC(C)(C)[C@@]1(OC(N)=O)CCCN(CC(=O)N2CCCC2)C1=O

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1L1 Q9UHC9 8/20 0.39
HTT P42858 1/20 0.38
CHRM2 P08172 5/20 0.34
CHRM4 P08173 4/20 0.34
CHRM1 P11229 4/20 0.34
CHRM3 P20309 4/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
GAA P10253 2/20 0.33
ALDH1A1 P00352 1/20 0.33
PRKCA P17252 1/20 0.33
GSK3B P49841 1/20 0.33
GFER P55789 1/20 0.32
MAPT P10636 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6984266 0.96 NPC1L1 (0.41) NPC1L1HTTCHRM2CHRM4CHRM1
SCHEMBL14677078 0.76 GRIN2B (0.34)
SCHEMBL7088438 0.75 TRPA1 (0.32) NPC1L1ALDH1A1
SCHEMBL7084911 0.74 GFER (0.46) CHRM2CHRM4CHRM1CHRM3ALDH1A1
SCHEMBL28702537 0.68 RXFP1 (0.34) HTTGAAALDH1A1MAPT
SCHEMBL15937080 0.64 GRIN2B (0.52) NPC1L1HTT
SCHEMBL5972238 0.62 F10 (0.42) CHRM2CHRM4CHRM1CHRM3ALDH1A1
SCHEMBL6982714 0.62 F10 (0.41) HTTCHRM2CHRM4CHRM1CHRM3
SCHEMBL6982717 0.62 F10 (0.41) HTTCHRM2CHRM4CHRM1CHRM3
SCHEMBL20407729 0.61 LMNA (0.39) NPC1L1HTTCHRM2CHRM4CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294716-A1 LACTAM INHIBITORS OF FACTOR XA AND METHOD Bristol-Myers Squibb Company (US) 2003-03-26 EP disclosed
WO-2001096331-A1 LACTAM INHIBITORS OF FACTOR XA AND METHOD BRISTOL-MYERS SQUIBB COMPANY (US) 2001-12-20 WO disclosed