SCHEMBL6982775

SCHEMBL6982775

CC(=O)Nc1c(C)c(C)c2c(c1C)CC(C)(CN1CCN(CCCCOC(c3ccccc3)c3ccccc3)CC1)O2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 5/20 0.37
SLC6A4 P31645 4/20 0.37
BCHE P06276 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
NFKB1 P19838 1/20 0.36
SLC6A2 P23975 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
THPO P40225 1/20 0.36
MTOR P42345 1/20 0.36
RAB9A P51151 1/20 0.36
HIF1A Q16665 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981136 0.87 SIGMAR1 (0.38) SLC6A3SLC6A4SMN1; SMN2TP53CYP1A2
Hydrochloric Acid SCHEMBL6979630 0.87 SMN1; SMN2 (0.39) SLC6A3SLC6A4SMN1; SMN2TP53CYP1A2
Hydrochloric Acid SCHEMBL6985051 0.83 SMN1; SMN2 (0.41) SLC6A3SLC6A4SMN1; SMN2TP53CYP1A2
Hydrochloric Acid SCHEMBL6985433 0.82 SMN1; SMN2 (0.41) SLC6A3SLC6A4SMN1; SMN2TP53CYP1A2
Hydrochloric Acid SCHEMBL6983996 0.82 SMN1; SMN2 (0.41) SLC6A3SLC6A4SMN1; SMN2TP53CYP1A2
SCHEMBL6983850 0.81 MEN1 (0.39) MAPTMEN1ALDH1A1LMNAKMT2A
Hydrochloric Acid SCHEMBL6985673 0.80 SMN1; SMN2 (0.42) SLC6A3SLC6A4SMN1; SMN2TP53CYP1A2
Hydrochloric Acid SCHEMBL6980238 0.80 ALDH1A1 (0.40) MAPTMEN1GMNNALDH1A1LMNA
SCHEMBL6985682 0.78 SLC6A4 (0.49) SLC6A3SLC6A4SLC6A2
SCHEMBL6980360 0.77 SLC18A3 (0.40) SMN1; SMN2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed