SCHEMBL6983805

SCHEMBL6983805

Fc1ccc(C(NC2CCNCC2)c2ccc(F)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 7/20 0.61
SLC6A2 P23975 7/20 0.61
SLC6A4 P31645 7/20 0.61
SLC6A3 Q01959 3/20 0.48
KCNH2 Q12809 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6030479 0.81 SOS1 (0.56) CHRM1SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL6984774 0.80 SOS1 (0.54) CHRM1SLC6A2SLC6A4
Bromide SCHEMBL7978275 0.80 SOS1 (0.54) CHRM1SLC6A2SLC6A4
Bromide SCHEMBL7978277 0.80 SOS1 (0.54) CHRM1SLC6A2SLC6A4
SCHEMBL8400412 0.79 HTR1D (0.43) CHRM1SLC6A2SLC6A4
SCHEMBL6979082 0.78 MAOA (0.51) CHRM1SLC6A2SLC6A4SLC6A3
SCHEMBL12715518 0.76 CHRM1 (1.00) CHRM1SLC6A2SLC6A4SLC6A3KCNH2
Propane SCHEMBL27576811 0.75 SOS1 (0.53) CHRM1SLC6A2SLC6A4
SCHEMBL377433 0.72 HTR6 (0.54) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7319671 0.72 SLC6A2 (0.45) SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed