SCHEMBL6984645

SCHEMBL6984645

Cc1ccc2cccc(NS(=O)(=O)c3ccccc3)c2n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC40A1 Q9NP59 8/20 1.00
GLO1 Q04760 3/20 1.00
AGTR1 P30556 3/20 1.00
PAX8 Q06710 2/20 1.00
TDP1 Q9NUW8 3/20 0.82
KMT2A Q03164 2/20 0.82
MEN1 O00255 1/20 0.82
NFKBIA P25963 6/20 0.67
RELA Q04206 5/20 0.67
MMP2 P08253 1/20 0.67
G6PD P11413 1/20 0.65
METAP2 P50579 1/20 0.65
METAP1 P53582 1/20 0.65
ATM Q13315 1/20 0.65
ALDH1A1 P00352 2/20 0.57
KDM4E B2RXH2 1/20 0.57
HPGD P15428 1/20 0.57
HSD17B10 Q99714 1/20 0.57
MITF O75030 1/20 0.57
S1PR4 O95977 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26053588 0.90 KMT2A (1.00) SLC40A1GLO1AGTR1PAX8TDP1
SCHEMBL23934032 0.85 KMT2A (0.76) SLC40A1GLO1AGTR1PAX8TDP1
SCHEMBL23934034 0.85 KMT2A (0.76) SLC40A1GLO1AGTR1PAX8TDP1
SCHEMBL22578645 0.84 KMT2A (0.74) SLC40A1GLO1AGTR1PAX8TDP1
SCHEMBL23933986 0.84 KMT2A (0.74) SLC40A1GLO1AGTR1PAX8TDP1
SCHEMBL2055432 0.83 SLC40A1 (0.71) SLC40A1GLO1AGTR1PAX8TDP1
SCHEMBL11973639 0.82 SLC40A1 (1.00) SLC40A1GLO1AGTR1PAX8TDP1
SCHEMBL23933988 0.82 TDP1 (0.71) SLC40A1GLO1AGTR1PAX8TDP1
SCHEMBL18889904 0.82 KMT2A (0.71) SLC40A1GLO1AGTR1PAX8TDP1
SCHEMBL11973111 0.81 SLC40A1 (1.00) SLC40A1GLO1AGTR1PAX8TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675526-B1 NOVEL SULFONAMINOQUINOLINE HEPCIDIN ANTAGONISTS VIFOR (INTERNATIONAL) AG (CH) 2017-02-01 EP disclosed
US-9102688-B2 Sulfonaminoquinoline hepcidin antagonists VIFOR (INTERNATIONAL) AG (CH) 2015-08-11 US disclosed
US-9102688-B2 Sulfonaminoquinoline hepcidin antagonists VIFOR (INTERNATIONAL) AG (CH) 2015-08-11 US disclosed
US-9102688-B2 Sulfonaminoquinoline hepcidin antagonists VIFOR (INTERNATIONAL) AG (CH) 2015-08-11 US disclosed
US-20140364424-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2014-12-11 US disclosed
US-20140364424-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2014-12-11 US disclosed
US-20140364424-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2014-12-11 US disclosed
CN-103492028-A Novel sulfonaminoquinoline hepcidin antagonists VIFOR INT AG 2014-01-01 CN disclosed
US-20120214803-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2012-08-23 US disclosed
US-20120214803-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2012-08-23 US disclosed
US-20120214803-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2012-08-23 US disclosed
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
US-6528187-B1 Luminescence element comprising pair of electrodes having formed therebetween plurality of organic compound thin film layers comprising electron-transporting layer which comprises specified compound FUJI PHOTO FILM CO., LTD. (JP) 2003-03-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120214803-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists HAMP, SLC40A1, FTH1 SLC40A1 2/4885GLO1 3935/4885AGTR1 2153/4885
US-20140364424-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists HAMP, SLC40A1, FTH1 SLC40A1 2/4885GLO1 3935/4885AGTR1 2153/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.